Associated Papers
Crystal structure of adenosine A2A receptor in complex with clinical candidate Etrumadenant reveals unprecedented antagonist interaction.
Claff T et al.
Communications Chemistry, 2023
37264098 (PubMed )
Supplement: 42004_2023_894_MOESM1_ESM.pdf
Dynamic behavior of the active and inactive states of the adenosine A(2A) receptor.
Lee S et al.
The Journal of Physical Chemistry. B, 2014
24579769 (PubMed )
Supplement: jp411618h_si_001.pdf
Arginine 199 and leucine 208 have key roles in the control of adenosine A2A receptor signalling function.
Bertheleme N et al.
Plos One, 2014
Loss of constitutive activity is correlated with increased thermostability of the human adenosine A2A receptor.
Bertheleme N et al.
British Journal of Pharmacology, 2013
Ligand-dependent activation and deactivation of the human adenosine A(2A) receptor.
Li J et al.
Journal of the American Chemical Society, 2013
Select a paper to view details